
个人简介
杨阳,讲师,男,1991.1, 2020年毕业与北京协和医学院(清华大学医学部),专业为药物化学,获医学博士学位,研究生导师:冯志强。
研究方向:抗肿瘤/小分子免疫治疗
代表性学术成果:
论文:
[1] Yang Y, Wang K, Chen H, et al. Design, synthesis, evaluation, and SAR of 4-phenylindoline derivatives, a novel class of small-molecule inhibitors of the programmed cell death-1/programmed cell death-ligand 1 (PD-1/PD-L1) interaction[J]. European Journal of Medicinal Chemistry, 2021, 211: 113001.
专利:
[1] Benzyl Phenyl Ether Derivative, Preparation Method Therefor, and Pharmaceutical Composition and Uses Thereof,WO2017202273A1, FENG Zhiqiang; CHEN Xiaoguang; YANG Yang; LAI Fangfang; JI Ming; ZHANG Lijing; ZHENG Yi; XUE Nina; WANG Ke; LI Ling.
[2] Nicotinyl Alcohol Ether Derivative, Preparation Method Therefor, and Pharmaceutical Composition and Uses Thereof, WO2017202274A1, FENG Zhiqiang; CHEN Xiaoguang; YANG Yang; ZHENG Yi; LAI Fangfang; JI Ming; ZHOU Chuan; ZHANG Lijing; WANG Ke; XUE Nina; LI Ling
[3] Bromo Benzyl Ether Derivative, Preparation Method Therefor, and Pharmaceutical Composition and Uses Thereof, WO2017202275A1, FENG Zhiqiang; CHEN Xiaoguang; ZHANG Lijing;YANG Yang; LAI Fangfang; JI Ming; ZHOU Chuan; ZHEN Yi; XUE Nina; LI Ling.
[4] Phenylate Derivative, Preparation Method Therefor, and Pharmaceutical Composition And Uses Thereof, WO2017202276A1, FENG Zhiqiang; CHEN Xiaoguang;YANG Yang; ZHOU Chuan; LAI Fangfang; JI Ming; JIN Xiaofeng; XUE Nina; ZHENG Yi; CHEN Hao; LI Ling.
[5]Method For Preparing 2-Hydroxyl-4-(2,3-Disubstituted Benzyloxy)-5-Substituted Benzaldehyde Derivative, WO2017202277A1, FENG Zhiqiang; CHEN Xiaoguang; YANG Yang; LAI Fangfang.
[6] 2-羟基-4-(2,3-双取代苄氧基)-5-取代苯甲醛衍生物的制备方法,CN107417506A, 冯志强; 陈晓光;杨阳; 来芳芳.
[7] 苄苯醚类衍生物、及其制法和药物组合物与用途,CN107417572A, 冯志强; 陈晓光; 杨阳; 来芳芳; 季鸣; 张莉婧; 郑义; 薛妮娜; 王克; 李凌.
[8] 烟醇醚类衍生物、及其制法和药物组合物与用途,CN109153670A, 冯志强; 陈晓光; 杨阳; 郑义; 来芳芳; 季鸣; 周川; 张莉婧; 王克; 薛妮娜; 李凌.
[9] 2-羟基-4-(2,3-双取代苄氧基)-5-取代苯甲醛衍生物的制备方法,CN109153626A, 冯志强; 陈晓光; 杨阳; 来芳芳.
[10] 苯醚类衍生物、及其制法和药物组合物与用途, CN109311792A, 冯志强; 陈晓光;杨阳;
周川; 来芳芳; 季鸣; 金小锋; 薛妮娜; 郑义; 陈浩; 李凌.
[11] 苯醚类衍生物、及其制法和药物组合物与用途,CN107417564A, 冯志强; 陈晓光;杨阳; 周川; 来芳芳; 季鸣; 金小锋; 薛妮娜; 郑义; 陈浩; 李凌.
[12] 溴代苄醚衍生物、及其制法和药物组合物与用途,CN107417666A, 冯志强; 陈晓光; 张莉婧; 杨阳; 来芳芳; 季鸣; 周川; 郑义; 薛妮娜; 李凌.
[13] 溴代苄醚衍生物、及其制法和药物组合物与用途,CN109195960A, 冯志强; 陈晓光; 张莉婧; 杨阳; 来芳芳; 季鸣; 周川; 郑义; 薛妮娜; 李凌.
[14] 碘同位素标记苄苯醚衍生物、及其制法和药物组合物与用途;CN111662270A; 冯志强,杨阳.
[15] 二氢吲哚衍生物、及其制法和药物组合物与用途;CN113444075A; 冯志强,杨阳.
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